TCS 401

CAS No. 243966-09-8

TCS 401 ( —— )

Catalog No. M20730 CAS No. 243966-09-8

TCS 401 is a selective inhibitor of protein-tyrosine phosphatase 1B (PTP1B; Ki = 0.29 μM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 58 In Stock
5MG 91 In Stock
10MG 146 In Stock
25MG 277 In Stock
50MG 464 In Stock
100MG 673 In Stock
200MG Get Quote In Stock
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Biological Information

  • Product Name
    TCS 401
  • Note
    Research use only not for human use.
  • Brief Description
    TCS 401 is a selective inhibitor of protein-tyrosine phosphatase 1B (PTP1B; Ki = 0.29 μM).
  • Description
    TCS 401 is a selective inhibitor of protein-tyrosine phosphatase 1B (PTP1B; Ki = 0.29 μM).
  • Synonyms
    ——
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    Phosphatase
  • Recptor
    PTP1B
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    243966-09-8
  • Formula Weight
    306.72
  • Molecular Formula
    C10H11ClN2O5S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:11 mg/mL (35.86 mM)
  • SMILES
    Cl.OC(=O)C(=O)Nc1sc2CNCCc2c1C(O)=O
  • Chemical Name
    2-(Oxaloamino)-4567-tetrahydrothieno[23-c]pyridine-3-carboxylic acid hydrochloride

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Du Z D Hu L T Zhao G Q et al. Protein tyrosine phosphatase 1B regulates the activity of retinal pigment epithelial cells[J]. Molecular vision 2015 21:523-531.
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